EXELIXIS, INC.; ANAND, Neel, Kumar; ARCALAS, Arlyn; BLAZEY, Charles, M.; BUHR, Chris, A.; CANNOY, Jonah; EPHSTEYN, Sergey; JOHNSON, Henry, William Beecroft; JOSHI, Anagha; KIM, Byung, Gyu; LEAHY, James, W.; LEE, Matthew, Sangyup; MA, Sunghoon; MAC, Morrison, B.; NUSS, John, M.; TAKEUCHI, Craig, Stacy; WANG, Longcheng; WANG, Yong Patent: WO2010/118208 A1, 2010 ; Location in patent: Page/Page column 250-251 ; WO 2010/118208 A1