BOEHRINGER INGELHEIM INTERNATIONAL GMBH; LLINAS-BRUNET, Montse; BORDELEAU , Josee; GODBOUT, Cedrickx; LEBLANC, Melissa; MOREAU, Benoit; O'MEARA, Jeffrey Patent: WO2011/63501 A1, 2011 ; Location in patent: Page/Page column 33 ; WO 2011/063501 A1