化学科研者一站式服务平台
-
地利洛非
Diprenorphine,17-(Cyclopropylmethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α,α-dimethyl-6,14-ethenomorphinan-7-methanol
化合物简介
Diprenorphine (brand name Revivon; former developmental code name M5050), also known as diprenorfin, is a non-selective, high-affinity, weak partial agonist of the μ- (MOR), κ- (KOR), and δ-opioid receptor (DOR) (with equal affinity) that is employed in veterinary medicine as an opioid antagonist. It is used to reverse the effects of super-potent opioid analgesics such as etorphine and carfentanil that are used for tranquilizing large animals. The drug is not approved for use in humans.
基本信息
CAS：14357-78-9
中文别名：利巴韦林杂质;
英文别名：DIPRENORPHINE;RX-5050M;Diprenorphin;DIPRENORPHINE POTENT OPIOID ANTAGON;diprenorpine;M-5050;
分子式：C26H35NO4
分子量：425.56
精确质量：425.257
Psa：62.16
Logp：3.3255
中文别名：利巴韦林杂质;
英文别名：DIPRENORPHINE;RX-5050M;Diprenorphin;DIPRENORPHINE POTENT OPIOID ANTAGON;diprenorpine;M-5050;
分子式：C26H35NO4
分子量：425.56
精确质量：425.257
Psa：62.16
Logp：3.3255
编号系统
UNII：1F0L5N25ZZ
物化性质
密度：1.33 g/cm3
折射率：1.656
折射率：1.656
安全信息
危险类别码：R20/21/22
危险品标志：Xn
危险品标志：Xn
生产方法及用途
合成路线
上游原料
下游产品
图谱
13C NMR : Predict
1H NMR : Predict
