MERCK SHARP and DOHME CORP.; KHAN, Tanweer; JOSIEN, Hubert; MCKITTRICK, Brian; VACCARO, Henry; BARA, Thomas; CALDWELL, John; HEAP, Charles, R.; GEISS, William, B.; MITRA, Surnya; ZYCH, Andrew, J. Patent: WO2013/142396 A1, 2013 ; Location in patent: Page/Page column 51 ;