JANSSEN PHARMACEUTICALS, INC.; CID-NUNEZ, Jose, Maria; TRABANCO-SUAREZ, Andres, Avelino; VEGA RAMIRO, Juan, Antonio; OEHLRICH, Daniel; TRESADERN, Gary, John; MACDONALD, Gregor, James Patent: WO2012/62759 A1, 2012 ; Location in patent: Page/Page column 47 ; WO 2012/062759 A1