FORMA THERAPEUTICS, INC.; BAIR, Kenneth W.; BUCKMELTER, Alexandre J.; HAN, Bingsong; LIN, Jian; REYNOLDS, Dominic J.; SMITH, Chase C.; WANG, Zhongguo; ZHENG, Xiaozhang Patent: WO2012/31199 A1, 2012 ; WO 2012/031199 A1