Merck Sharp & Dohme Corp.; DENG, Yongqi; CURRAN, Patrick, J.; SHIPPS, Gerald W., Jr.; ZHAO, Lianyun; SIDDIQUI, M. Arshad; POPOVICI-MULLER, Janeta; DUCA, Jose, S.; HRUZA, Alan, W.; FISCHMANN, Thierry, O.; MADISON, Vincent, S.; ZHANG, Rumin; MCNEMAR, Charles, Wayne; MAYHOOD, Todd, W.; WINDSOR, William, T.; LEES, Emma, M.; PARRY, David, A. Patent: EP1931657 B1, 2013