BRISTOL-MYERS SQUIBB COMPANY; AHMAD, Saleem; WASHBURN, William, N.; HERNANDEZ, Andres, S.; ROBL, Jeffrey, A.; NGU, Khehyong; WANG, Zhenghua Patent: WO2010/104830 A1, 2010 ; Location in patent: Page/Page column 70-71 ; WO 2010/104830 A1