Janssen Pharmaceuticals, Inc.; Andrés-Gil, José Ignacio; Alcázar-Vaca, Manuel Jesús; Cid-Núñez, José Maria; Trabanco-Suárez, Andrés Avelino; Bormans, Guy Maurits R.; Celen, Sofie Jeanne Leopoldine; Koole, Michel Patent: US2013/230459 A1, 2013 ; Location in patent: Paragraph 0154 ;