Pautus, Stephane; Sehr, Peter; Lewis, Joe; Fortune, Antoine; Wolkerstorfer, Andrea; Szolar, Oliver; Guilligay, Delphine; Lunardi, Thomas; Decout, Jean-Luc; Cusack, Stephen Journal of Medicinal Chemistry, 2013 , vol. 56, # 21 p. 8915 - 8930