SANOFI-AVENTIS; GESSLER, Simon; GILL, Harpal S.; LEE, George E.; PLETTENBURG, Oliver; PODESCHWA, Michael; POWERS, Matthew R.; ROSSEN, Kai; SHRIMP, II, Frederick L.; SUBOTKOWSKI, Witold; VANASSE, Benoit J.; WEHLAN, Hermut A.; WEIBERTH, Franz J.; YU, Yong; ZHANG, Jiuqing Patent: WO2010/77623 A1, 2010 ; Location in patent: Page/Page column 53 ;