ELI LILLY AND COMPANY; DODGE, Jeffrey, Alan; RICHARDSON, Timothy, Ivo; CLARKE, Christian, Alexander; JONES, Scott, Alan; HINKLIN, Ronald, Jay; HUMMEL, Conrad, Wilson; LEWIS, George, Sal Patent: WO2010/36497 A2, 2010 ; Location in patent: Page/Page column 53; 54; 55 ;