WYETH LLC; AYRAL-KALOUSTIAN, Semiramis; MANSOUR, Tarek Suhayl; TSOU, Hwei-Ru; ZHANG, Nan; VENKATESAN, Aranapakam M.; DI, Li; KERNS, Edward H. Patent: WO2010/30727 A1, 2010 ; Location in patent: Page/Page column 98 ; WO 2010/030727 A1