N.V. ORGANON; PHARMACOPEIA, LLC; PALIN, Ronald; RATCLIFFE, Paul, David; KULTGEN, Steven, G.; HO, Koc-Kan; ROUGHTON, Andrew, Laird; OHLMEYER, Michael Patent: WO2010/91009 A1, 2010 ; Location in patent: Page/Page column 41 ; WO 2010/091009 A1