BRISTOL-MYERS SQUIBB COMPANY; PURANDARE, Ashok V.; FRENNESSON, David B.; KAMAU, Muthoni G.; HARIKRISHNAN, Lalgudi S.; SAULNIER, Mark G. Patent: WO2010/42684 A1, 2010 ; Location in patent: Page/Page column 58 ; WO 2010/042684 A1