Orrling, Kristina M.; Jansen, Chimed; Vu, Xuan Lan; Balmer, Vreni; Bregy, Patrick; Shanmugham, Anitha; England, Paul; Bailey, David; Cos, Paul; Maes, Louis; Adams, Emily; Van Den Bogaart, Erika; Chatelain, Eric; Ioset, Jean-Robert; Van De Stolpe, Andrea; Zorg, Stephanie; Veerman, Johan; Seebeck, Thomas; Sterk, Geert Jan; De Esch, Iwan J. P.; Leurs, Rob Journal of Medicinal Chemistry, 2012 , vol. 55, # 20 p. 8745 - 8756