MERCK SHARP and DOHME CORP.; ALI, Amjad; BENNETT, D. Jonathan; CAI, Jaiqiang; CARSWELL, Emma; COOKE, Andrew; HOYT, Scott, B.; LO, Michael; LONDON, Clare; MACLEAN, John; PARK, Min, K.; RATCLIFFE, Paul; TAYLOR, Jerry Andrew; WHITEHEAD, Brent; XIONG, Yusheng Patent: WO2013/43518 A1, 2013 ; Location in patent: Page/Page column 36 ;