Rai, Ganesha; Sayed, Ahmed A.; Lea, Wendy A.; Luecke, Hans F.; Chakrapani, Harinath; Prast-Nielsen, Stefanie; Jadhav, Ajit; Leister, William; Shen, Min; Inglese, James; Austin, Christopher P.; Keefer, Larry; Arner, Elias S. J.; Simeonov, Anton; Maloney, David J.; Williams, David L.; Thomas, Craig J. Journal of Medicinal Chemistry, 2009 , vol. 52, # 20 p. 6474 - 6483