BRISTOL-MYERS SQUIBB COMPANY; LEXICON PHARMACEUTICALS, INC.; BI, Yingzhi; DZIERBA, Carolyn, Diane; BRONSON, Joanne, J.; FINK, Cynthia; GREEN, Michael; KIMBALL, David; MACOR, John, E.; KWON, Soojin; ZHANG, Yulian; ZIPP, Greg Patent: WO2011/44212 A1, 2011 ; Location in patent: Page/Page column 30-31 ;