MERCK SHARP and DOHME CORP.; COLEMAN, Paul, J.; EMBREY, Mark; HARTINGH, Timothy, J.; POWELL, David; RAHEEM, Izzat, T.; CHANG, Ronald, K.; SCHREIER, John; SISKO, John; STEELE, Tom; WALJI, Abbas Patent: WO2014/18449 A1, 2014 ; Location in patent: Page/Page column 36 ;