Wakenhut, Florian; Tran, Thien Duc; Pickford, Chris; Shaw, Stephen; Westby, Mike; Smith-Burchnell, Caroline; Watson, Lesa; Paradowski, Michael; Milbank, Jared; Stonehouse, David; Cheung, Kathy; Wybrow, Robert; Daverio, Felice; Crook, Samuel; Statham, Keith; Leese, David; Stead, Darren; Adam, Fiona; Hay, Duncan; Roberts, Lee R.; Chiva, Jean-Yves; Nichols, Carly; Blakemore, David C.; Goetz, Gilles H.; Che, Ye; Gardner, Iain; Dayal, Satish; Pike, Andrew; Webster, Rob; Pryde, David C. ChemMedChem, 2014, vol. 9, # 7 p. 1387 - 1396 doi: 10.1002/cmdc.201400046