JANSSEN PHARMACEUTICALS, INC.; DEPRÉ, Dominique Paul Michel; ORMEROD, Dominic John; HORVATH, Andras; MOODY, Thomas Shaw; BROSSAT, Maude; RIANT, Olivier; VRIAMONT, Nicolas; LEMAIRE, Sébastien François Emmanuel; HERMANT, Sébastien Nicolas J Patent: WO2016/157058 A1, 2016