RFS PHARMA, LLC; SCHINAZI, Raymond, F.; MELLORS, John, W.; SLUIS-CREMER, Nicolas, Paul; AMBLARD, Frank; COATS, Steven, J.; SHI, Junxing; WHITAKER, Richard, Anthony; EMORY UNIVERSITY; UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION Patent: WO2010/68708 A2, 2010