VANDERBILT UNIVERSITY; JANSSEN PHARMACEUTICA NV; JANSSEN-CILAG SA; CONN, P., Jeffrey; LINDSLEY, Craig, W.; STAUFFER, Shaun, R.; JONES, Carrie, K.; BARTOLOME-NEBREDA, Jose, Manuel; CONDE-CEIDE, Susana; MACDONALD, Gregor, James; ALCAZAR VACA, Manuel, Jesus Patent: WO2012/31024 A1, 2012