ORCHID PHARMA LTD.; MERCK SHARP & DOHME CORP.; BALASUBRAMANIAN, Gopalan; PAUL-SATYASEELA, Maneesh; SRINIVASAN, Chidambaram, Venkateswaran; LYER, Sridhar, Ramanathan; PERIASAMY, Hariharan; PARAMESWARAN, Venkatesan; THIRUNAVUKKARASU, Bharani; GUNTURU, Prabhakar, Rao; DESHKUMAR, Manjula, Devi; JAKKALA, Venkateshwarlu; NARGUND, Ravi, P.; MILLER, Michael; SINGH, Sheo; DONG, Shuzhi; WANG, Hongwu; YOUNG, Katherine Patent: WO2017/158616 A1, 2017