EPIZYME, INC.; OLHAVA, Edward, James; CHESWORTH, Richard; KUNTZ, Kevin, Wayne; RICHON, Victoria, Marie; POLLOCK, Roy, Macfarlane; DAIGLE, Scott, Richard Patent: WO2012/75381 A1, 2012 ; Location in patent: Page/Page column 210 ; WO 2012/075381 A1