Mirguet, Olivier; Gosmini, Romain; Toum, Jeroime; Clement, Catherine A.; Barnathan, Melanie; Brusq, Jean-Marie; Mordaunt, Jacqueline E.; Grimes, Richard M.; Crowe, Miriam; Pineau, Olivier; Ajakane, Myriam; Daugan, Alain; Jeffrey, Phillip; Cutler, Leanne; Haynes, Andrea C.; Smithers, Nicholas N.; Chung, Chun-Wa; Bamborough, Paul; Uings, Iain J.; Lewis, Antonia; Witherington, Jason; Parr, Nigel; Prinjha, Rab K.; Nicodeme, Edwige Journal of Medicinal Chemistry, 2013, vol. 56, # 19 p. 7501 - 7515 doi: 10.1021/jm401088k