Kawamura, Shuhei; Ito, Yoshihiko; Hirokawa, Takatsugu; Hikiyama, Eriko; Yamada, Shizuo; Shuto, Satoshi Journal of Medicinal Chemistry, 2018, vol. 61, # 9 p. 4020 - 4029 doi: 10.1021/acs.jmedchem.8b00041