MERCK SHARP and DOHME CORP.; BENNETT, Frank; HUANG, Yuhua; WANG, Lingyan; BOGEN, Stephane, L.; KEREKES, Angela, D.; GIRIJAVALLABHAN, Vinay M.; BUTORA, Gabor; TRUONG, Quang; DAVIES, Ian; WEBER, Anne E. Patent: WO2014/78463 A1, 2014 ;