Eisai RandD Management Co., Ltd.; CLARK, Richard; MATSUURA, Fumiyoshi; SHINODA, Masanobu; HIROTA, Shinsuke; KIRA, Kazunobu; AZUMA, Hiroshi; TAKEMURA, Atsushi; YASUI, So; KUSANO, Kazutomi; MIKAMOTO, Masaki; OMAE, Takao Patent: WO2011/145747 A1, 2011 ; Location in patent: Page/Page column 97-98 ; WO 2011/145747 A1