TETRAPHASE PHARMACEUTICALS, INC.; ZHOU, Jingye; XIAO, Xiao-Yi; PLAMONDON, Louis; HUNT, Diana, Katharine; CLARK, Roger, B.; ZAHLER, Robert, B. Patent: WO2010/17470 A1, 2010 ; Location in patent: Page/Page column 113-115 ; WO 2010/017470 A1