ARRAY BIOPHARMA INC.; GENENTECH, INC.; ALIAGAS, Ignacio; GRADL, Stefan; GUNZNER, Janet; MATHIEU, Simon; RUDOLPH, Joachim; WEN, Zhaoyang; WENGLOWSKY, Steven Mark Patent: WO2011/25947 A1, 2011 ; Location in patent: Page/Page column 44 ; WO 2011/025947 A1