Ann, Jihyae; Czikora, Agnes; Saini, Amandeep S.; Zhou, Xiaoling; Mitchell, Gary A.; Lewin, Nancy E.; Peach, Megan L.; Blumberg, Peter M.; Lee, Jeewoo Journal of Medicinal Chemistry, 2018, vol. 61, # 14 p. 6261 - 6276 doi: 10.1021/acs.jmedchem.8b00661